Test
Inhibits NF-κB activation
CaM kinase II inhibitor; water soluble version of KN 93 (Cat. No. 1278).
Highly potent PORCN inhibitor
Selective Mps1 kinase inhibitor
High affinity, potent and selective Hsp90 inhibitor
Potent non-peptide oxytocin receptor partial agonist; also V1a receptor antagonist
Non-selective P2 agonist; analog of ATP (Cat. No. 3245)
High affinity, selective urotensin II (UT) receptor antagonist
Potent PORCN inhibitor; active in vivo
Selective inducer of neuronal differentiation in hippocampal neural progenitors
gp130 inhibitor; blocks cytokine-triggered gp130 signaling
HECT E3 ubiquitin ligase inhibitor
Potent IR and IGF1R inhibitor; also inhibits anaplastic lymphoma kinase (ALK)
Selective DDR1 inhibitor
Potent and selective PERK inhibitor; orally bioavailable