Test
Competitive serine protease inhibitor
Broad spectrum, irreversible inhibitor of serine proteases
Potent and selective negative allosteric modulator at mGlu1; also mGlu1 inverse agonist
MEK inhibitor
Antimicrobial peptide derivative of human cathelicidin
Selective inhibitor of Rac1-GEF interaction; antioncogenic
Selective FFA4 (GPR120) antagonist
High affinity Smurf1 inhibitor; enhances BMP signaling
Potent and selective LDHA inhibitor
Highly potent and selective JNK3 inhibitor
Highly selective and potent non-peptide NPY Y5 receptor antagonist
BET bromodomain inhibitor; arrests cell cycle at G1 phase
Potent and selective K2P3.1 (TASK-1) channel blocker
Potent and selective Lck and Src inhibitor; also inhibits SIK
Glucokinase activator